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Dr. Sunil K. Upadhyay
Dr. Sunil K. Upadhyay
Verified email at thermofisher.com - Homepage
Title
Cited by
Cited by
Year
Conversion of abiraterone to D4A drives anti-tumour activity in prostate cancer
RJANS Zhenfei Li, Andrew C. Bishop, Mohammad Alyamani, Jorge A. Garcia ...
Nature 523 (7560), 347-351, 2015
2852015
Adrenal-derived 11-Oxygenated 19-Carbon Steroids are the Dominant Androgens in Classic 21-Hydroxylase Deficiency
AFTATNRCSKUTGJJSDPMWRR Auchus
European Journal of Endocrinology 174, 601-609, 2016
2042016
Redirecting abiraterone metabolism to biochemically fine tune prostate cancer anti-androgen therapy
NS Zhenfei Li, Mohammad Alyammani, Jianneng Li, Kevin Rogacki, Mohamed ...
Nature 533, 547-551, 2016
1672016
High-affinity small-molecule inhibitors of the menin-mixed lineage leukemia (MLL) interaction closely mimic a natural protein–protein interaction
S He, TJ Senter, J Pollock, C Han, SK Upadhyay, T Purohit, RD Gogliotti, ...
Journal of medicinal chemistry 57 (4), 1543-1556, 2014
1112014
Steroidogenic Metabolism of Galeterone Reveals a Diversity of Biochemical Activities
RJANS Mohammad Alyamani,Zhenfei Li,Michael Berk,Jianneng Li, Jingjie Tang ...
Cell Chemical Biology 24, 825-832, 2017
502017
HSD3B1(1245A>C) variant regulates dueling abiraterone metabolite effects in prostate cancer
M Alyamani, H Emamekhoo, S Park, J Taylor, N Almassi, S Upadhyay, ...
The Journal of clinical investigation 128 (8), 3333-3340, 2018
492018
A-ring modified steroidal azoles retaining similar potent and slowly reversible CYP17A1 inhibition as abiraterone
M Garrido, HM Peng, FK Yoshimoto, SK Upadhyay, E Bratoeff, RJ Auchus
The Journal of steroid biochemistry and molecular biology 143, 1-10, 2014
382014
Comparison of microwave-assisted and conventional preparations of cyclic imides
SK Upadhyay, SRK Pingali, BS Jursic
Tetrahedron Letters 51 (17), 2215-2217, 2010
382010
Development and Validation of a Novel LC-MS/MS Method for Simultaneous Determination of Abiraterone and Its Seven Metabolites in Human Serum: Innovation in Separation of …
MAZLSKUDARJAN Sharifi
Journal of Steroidal Biochemistry and Molecular Biology 172, 231-239, 2017
31*2017
Microwave-assisted benzyl mono-and dibromination in diethyl carbonate as environmentally friendly alternative to radical bromination in carbon tetrachloride
SRK Pingali, SK Upadhyay, BS Jursic
Green chemistry 13 (4), 928-933, 2011
262011
menin-MLL inhibitors and methods of use thereof
TJS Jolanta Grembecka, Tomasz Cierpicki, Sunil Kumar Upadhyay, Shaun R ...
WO Patent WO 2014200479 A1 20,141,218, 2014
20*2014
Novel and efficient synthesis and antifungal evaluation of 2, 3-functionalized cholestane and androstane derivatives
BS Jursic, SK Upadhyay, CC Creech, DM Neumann
Bioorganic & medicinal chemistry letters 20 (24), 7372-7375, 2010
192010
Visible-Light-Driven Oxidative Mono-and Dibromination of Benzylic sp3 C–H Bonds with Potassium Bromide/Oxone at Room Temperature
M Zhao, M Li, W Lu
Synthesis 50 (24), 4933-4939, 2018
162018
Afatinib use in non-small cell lung cancer previously sensitive to epidermal growth factor receptor inhibitors: The United Kingdom Named Patient Programme
F Khan, C Ottensmeier, S Popat, D Dua, N Dorey, S Ellis, M Szabo, ...
European journal of cancer 50 (10), 1717-1721, 2014
152014
Synthesis and antifungal activity of functionalized 2, 3-spirostane isomers
SK Upadhyay, CC Creech, KL Bowdy, ED Stevens, BS Jursic, ...
Bioorganic & medicinal chemistry letters 21 (10), 2826-2831, 2011
152011
Antifungal activity of 2α, 3β-functionalized steroids stereoselectively increases with the addition of oligosaccharides
A Cammarata, SK Upadhyay, BS Jursic, DM Neumann
Bioorganic & medicinal chemistry letters 21 (24), 7379-7386, 2011
92011
Sulfur Betaines from S-Propargyl Xanthates. Unusual Chemistry from a Simple Functional Group
SZ Zard
Synthesis 51 (05), 1006-1020, 2019
62019
HSD3B1 genotype and abiraterone (Abi) metabolites in patients (pts) with prostate cancer (PCa).
H Emamekhoo, M Alyamani, S Park, J Taylor, N Almassi, S Upadhyay, ...
Journal of Clinical Oncology 36 (6_suppl), 325-325, 2018
52018
Microwave-Assisted NBS Bromination of p-Iminotoluenes: Preparation of New Alcohol, Mercapto, and Amino Protection Groups
SK Upadhyay, BS Jursic
Synthetic Communications 41 (21), 3177-3185, 2011
42011
A socio-economic analysis of fish farming in Gonda and Basti districts, Uttar Pradesh.
SK Upadhyay, J Mishra
22020
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